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Home - Products - GPCR/G Protein - 5-HT Receptor - WAY-100635 maleate (b)

WAY-100635 maleate (b)

CAS No. 634908-75-1

WAY-100635 maleate (b)( WAY 100635 maleate salt | WAY100635 maleate salt )

Catalog No. M15399 CAS No. 634908-75-1

WAY-100635 is a potent and selective 5-HT1A receptor antagonist; also acts as potent full agonist at the D4 receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 34 In Stock
5MG 55 In Stock
10MG 86 In Stock
25MG 146 In Stock
50MG 214 In Stock
100MG 317 In Stock
500MG 764 In Stock
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Biological Information

  • Product Name
    WAY-100635 maleate (b)
  • Note
    Research use only, not for human use.
  • Brief Description
    WAY-100635 is a potent and selective 5-HT1A receptor antagonist; also acts as potent full agonist at the D4 receptor.
  • Description
    WAY-100635 is a potent and selective 5-HT1A receptor antagonist; also acts as potent full agonist at the D4 receptor; completely prevents not only the hyperpolarization, with an IC50 of 1.3 nM, but also the decrease in membrane input resistance produced by 5-HT and 5-carboxamidotryptamine with IC50 of 22.5 μM and 50 nM, respectively.Anxiety Phase 1 Discontinued.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    WAY 100635 maleate salt | WAY100635 maleate salt
  • Pathway
    GPCR/G Protein
  • Target
    5-HT Receptor
  • Recptor
    5-HT1A
  • Research Area
    Neurological Disease
  • Indication
    Anxiety

Chemical Information

  • CAS Number
    634908-75-1
  • Formula Weight
    538.6352
  • Molecular Formula
    C29H38N4O6
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO: ≥ 34 mg/mL
  • SMILES
    COC1=CC=CC=C1N2CCN(CC2)CCN(C3=CC=CC=N3)C(=O)C4CCCCC4.C(=CC(=O)O)C(=O)O
  • Chemical Name
    Cyclohexanecarboxamide, N-[2-[4-(2-methoxyphenyl)-1-piperazinyl]ethyl]-N-2-pyridinyl-, (2Z)-2-butenedioate (9CI)

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Corradetti R, et al. J Pharmacol Exp Ther. 1996 Aug;278(2):679-88. 2. Fornal CA, et al. J Pharmacol Exp Ther. 1996 Aug;278(2):752-62. 3. García G, et al. Eur J Med Chem. 2014 Oct 6;85:795-806.
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